HCA ISOENZYME INHIBITORY ACTIVITIES OF SCHIFF BASES DERIVED FROM CINNAMALDEHYDE AND P-METHOXYCINNAMALDEHYDE


Celik H., Maman M., Babagil A.

FRESENIUS ENVIRONMENTAL BULLETIN, cilt.27, sa.6, ss.4469-4482, 2018 (SCI-Expanded, Scopus)

  • Yayın Türü: Makale / Tam Makale
  • Cilt numarası: 27 Sayı: 6
  • Basım Tarihi: 2018
  • Dergi Adı: FRESENIUS ENVIRONMENTAL BULLETIN
  • Derginin Tarandığı İndeksler: Science Citation Index Expanded (SCI-EXPANDED), Scopus
  • Sayfa Sayıları: ss.4469-4482
  • Atatürk Üniversitesi Adresli: Evet

Özet

In this study, eight different Schiff base derivatives, derived from cinnamaldehyde and p-methoxycinnamaldehyde were synthesized from the corresponding cinnamaldehydes and anilines via microwave irradiation and their inhibition of activity on the hCA-I and hCA-II isoenzymes were investigated. IC50 values of seven compounds showed to have more stronger inhibitor effects than the reference inhibitor acetazolamide.